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Youbo Zhang1,2,Tingting Yan2,Tianxia Wang1,3,Xiaoyan Liu1,Keisuke Hamada2,Dongxue Sun2,Yizheng Sun1,Yanfang Yang1,Jing Wang1,Shogo Takahashi2,Qiong Wang2,Kristopher W.Krausz2,Changtao Jiang4,Cen Xie2,Xiuwei Yang1,Frank J.Gonzalez2(State Key Laboratory of Natural and Biomimetic Drugs and Department of Natural Medicines,School of Pharmaceutical Sciences,Peking University;Laboratory of Metabolism,Center for Cancer Research,National Cancer Institute,National Institutes of Health;School of Life Science and Engineering,Lanzhou University of Technology;Department of Physiology and Pathophysiology,School of Basic Medical Sciences,Peking University,the Key Laboratory of Molecular Cardiovascular Science,Ministry of Education).Crosstalk between CYP2E1 and PPARα substrates and agonists modulate adipose browning and obesity[J].Acta Pharmaceutica Sinica B,2022,第5期
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Abi Maharjan1,2,3,Hongyu Sun1,4,Zeying Cao1,3,Ke Li3,5,Jinping Liu6,Jun Liu1,7,Tiqiao Xiao5,Guanyun Peng5,Junqiu Ji7,Peter York1,Balmukunda Regmi8,Xianzhen Yin1,7,Jiwen Zhang1,3,4,Li Wu1,2(Center for Drug Delivery System,Shanghai Institute of Materia Medica,Chinese Academy of Sciences;School of Pharmacy,Key Laboratory of Molecular Pharmacology and Drug Evaluation,Ministry of Education,Yantai University;University of Chinese Academy of Sciences;NMPA Key Laboratory for Quality Research and Evaluation of Pharmaceutical Excipients,National Institutes for Food and Drug Control;Shanghai Synchrotron Radiation Facility/Zhangjiang Lab,Shanghai Advanced Research Institute,Chinese Academy of Sciences;Hefei Lifeon Medication Group;Center for MOST and Image Fusion Analysis,Shanghai Institute of Materia Medica,Chinese Academy of Sciences;Maharajgung Medical Campus,Institute of Medicine,Tribhuvan University).Redefinition to bilayer osmotic pump tablets as subterranean river system within mini-earth via three-dimensional structure mechanism[J].Acta Pharmaceutica Sinica B,2022,第5期
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Elisa Rioja-Blanco1,2,Irene Arroyo-Solera1,2,3,Patricia álamo1,2,3,Isolda Casanova1,2,3,Alberto Gallardo1,4,Ugutz Unzueta1,2,3,Naroa Serna3,5,6,Laura Sánchez-García3,5,6,Miquel Quer3,7,Antonio Villaverde3,5,6,Esther Vázquez3,5,6,Ramon Mangues1,2,3,Lorena Alba-Castellón1,2,Xavier León3,7(Institut d'Investigació Biomèdica Sant Pau(IIB-Sant Pau) Institut de Recerca contra la Leucèmia Josep Carreras CIBER de Bioingeniería,Biomateriales y Nanomedicina(CIBER-BBN);Department of Pathology,Hospital de la Santa Creu i Sant Pau;Institut de Biotecnologia i de Biomedicina,Universitat Autònoma de Barcelona;Departament de Genètica i de Microbiologia,Universitat Autònoma de Barcelona;Department of Otorhinolaryngology,Hospital de la Santa Creu i Sant Pau).Self-assembling protein nanocarrier for selective delivery of cytotoxic polypeptides to CXCR4+ head and neck squamous cell carcinoma tumors[J].Acta Pharmaceutica Sinica B,2022,第5期
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Zhuo-Xun Wu1,Qiu-Xu Teng1,Yuqi Yang1,Nikita Acharekar1,Jing-Quan Wang1,Min He2,Sabesan Yoganathan1,Jun Lin3,Jian Wang2,Zhe-Sheng Chen1(Department of Pharmaceutical Sciences,College of Pharmacy and Health Sciences,St.John's University;Department of Radiotherapy,the Affiliated Jiangyin People's Hospital of Nantong University;Department of Anesthesiology,Stony Brook University Health Sciences Center).MET inhibitor tepotinib antagonizes multidrug resistance mediated by ABCG2 transporter:In vitro and in vivo study[J].Acta Pharmaceutica Sinica B,2022,第5期
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Jie Chang1,2,Ruirui Yang2,3,4,Lifan Chen2,3,Zisheng Fan1,2,Jingyi Zhou1,2,Hao Guo2,3,Yinghui Zhang2,3,Yadan Liu1,2,Guizhen Zhou1,2,Keke Zhang1,2,Kaixian Chen2,3,1,Hualiang Jiang2,3,1,4,Mingyue Zheng2,3,1,Sulin Zhang2,3(School of Chinese Materia Medica,Nanjing University of Chinese Medicine;Drug Discovery and Design Center,State Key Laboratory of Drug Research,Shanghai Institute of Materia Medica,Chinese Academy of Sciences;University of Chinese Academy of Sciences;Shanghai Institute for Advanced Immunochemical Studies,and School of Life Science and Technology,ShanghaiTech University).Discovery of ARF1-targeting inhibitor demethylzeylasteral as a potential agent against breast cancer[J].Acta Pharmaceutica Sinica B,2022,第5期
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Editoral Office of Acta Pharmaceutica Sinica(Editoral Office of Acta Pharmaceutica Sinica).Information for Authors[J].Acta Pharmaceutica Sinica B,2022,第5期
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Guangdi Li1,Yali Wang1,Erik De Clercq2(Hunan Provincial Key Laboratory of Clinical Epidemiology,Xiangya School of Public Health,Central South University;Rega Institute for Medical Research,Department of Microbiology,Immunology and Transplantation).Approved HIV reverse transcriptase inhibitors in the past decade[J].Acta Pharmaceutica Sinica B,2022,第4期
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Minyang Fu,Dandan Peng,Tianxia Lan,Yuquan Wei,Xiawei Wei(Laboratory of Aging Research and Cancer Drug Target,State Key Laboratory of Biotherapy,National Clinical Research Center for Geriatrics,West China Hospital,Sichuan University).Multifunctional regulatory protein connective tissue growth factor(CTGF):A potential therapeutic target for diverse diseases[J].Acta Pharmaceutica Sinica B,2022,第4期
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Tiecheng Zhong,Wenxin Zhang,Hongjie Guo,Xiaohui Pan,Xi Chen,Qiaojun He,Bo Yang,Ling Ding(Zhejiang Province Key Laboratory of Anti-Cancer Drug Research,Institute of Pharmacology and Toxicology,College of Pharmaceutical Sciences,Zhejiang University).The regulatory and modulatory roles of TRP family channels in malignant tumors and relevant therapeutic strategies[J].Acta Pharmaceutica Sinica B,2022,第4期
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Pengcheng Wang1,2,3,Guangyi Zeng1,2,3,Yu Yan1,3,Song-yang Zhang1,3,Yongqiang Dong1,3,Yangming Zhang1,3,Xingzhong Zhang1,3,Huiying Liu1,3,Zhipeng Zhang4,Changtao Jiang1,2,3,Yanli Pang5(Department of Physiology and Pathophysiology,School of Basic Medical Sciences,Peking University,Key Laboratory of Molecular Cardiovascular Science,Ministry of Education;Center of Basic Medical Research,Institute of Medical Innovation and Research,Peking University Third Hospital;Center for Obesity and Metabolic Disease Research,School of Basic Medical Sciences,Peking University;General Surgery Department,Peking University Third Hospital;Center for Reproductive Medicine,Department of Obstetrics and Gynecology,Peking University Third Hospital).Disruption of adipocyte HIF-1α improves atherosclerosis through the inhibition of ceramide generation[J].Acta Pharmaceutica Sinica B,2022,第4期
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Hui Liu1,Weimin Qiu1,Tianyu Sun1,Lei Wang1,Chenxi Du1,Yanyu Hu2,Wenyuan Liu1,3,Feng Feng4,2,Yao Chen5,Haopeng Sun1,4(School of Pharmacy,China Pharmaceutical University;Department of Natural Medicinal Chemistry,China Pharmaceutical University;Department of Pharmaceutical Analysis,Key Laboratory of Drug Quality Control and Pharmacovigilance,China Pharmaceutical University;Jiangsu Drug Development Engineering Research Center for Central Degenerative Disease,Jiangsu Food and Pharmaceuticals Science College;School of Pharmacy,Nanjing University of Chinese Medicine).Therapeutic strategies of glioblastoma(GBM):The current advances in the molecular targets and bioactive small molecule compounds[J].Acta Pharmaceutica Sinica B,2022,第4期
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Lingxin Hou1,Ying Zhang1,Han Ju1,Srinivasulu Cherukupalli1,Ruifang Jia1,Jian Zhang2,Bing Huang3,Arianna Loregian4,Xinyong Liu1,5,Peng Zhan1,5(Department of Medicinal Chemistry,Key Laboratory of Chemical Biology(Ministry of Education),School of Pharmaceutical Sciences,Cheeloo College of Medicine,Shandong University;Institute of Medical Sciences,The Second Hospital,Cheeloo College of Medicine,Shandong University;Institute of Poultry Science,Shandong Academy of Agricultural Sciences;Department of Molecular Medicine,University of Padova;China-Belgium Collaborative Research Center for Innovative Antiviral Drugs of Shandong Province).Contemporary medicinal chemistry strategies for the discovery and optimization of infiuenza inhibitors targeting vRNP constituent proteins[J].Acta Pharmaceutica Sinica B,2022,第4期
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Songli Wang1,2,Ruifeng Wang1,Nana Meng1,Linwei Lu3,Jun Wang1,Jianfen Zhou1,Jiasheng Lu1,Qianzhu Xu1,Cao Xie1,Changyou Zhan1,2,Yao Li4,Yang Yu4,Weiyue Lu1,5,6,Min Liu1(Department of Pharmaceutics,School of Pharmacy,Key Laboratory of Smart Drug Delivery(Ministry of Education and PLA),Fudan University;Department of Pharmacology,School of Basic Medical Sciences,Fudan University;The Department of Integrative Medicine,Huashan Hospital,Fudan University and the Institutes of Integrative Medicine of Fudan University;The National Facility for Protein Science in Shanghai(NFPS);State Key Laboratory of Medical Neurobiology and the Collaborative Innovation Center for Brain Science and Department of Pharmacology,School of Basic Medical Sciences,Fudan University;Minhang Branch,Zhongshan Hospital and Institute of Fudan-Minhang Academic Health System,Minhang Hospital,Fudan University).Engineered platelets-based drug delivery platform for targeted thrombolysis[J].Acta Pharmaceutica Sinica B,2022,第4期
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Mengqi Xu1,Cong Mao2,Haoting Chen2,Lu Liu3,Yabin Wang1,Abid Hussain3,Sulei Li1,Xu Zhang4,Ruslan G.Tuguntaev2,Xing-Jie Liang3,Weisheng Guo2,Feng Cao1(Department of Cardiology,National Clinical Research Center for Geriatric Diseases&Second Medical Center of Chinese PLA General Hospital;Department of Minimally Invasive Interventional Radiology,Key Laboratory of Molecular Target&Clinical Pharmacology,School of Pharmaceutical Sciences&the Second Affiliated Hospital,Guangzhou Medical University;Laboratory of Controllable Nanopharmaceuticals,Chinese Academy of Sciences(CAS)Center for Excellence in Nanoscience and CAS Key Laboratory for Biomedical Effects of Nanomaterials and Nanosafety,National Center for Nanoscience and Technology;Department of Urology,Chinese PLA General Hospital).Osteopontin targeted theranostic nanoprobes for laser-induced synergistic regression of vulnerable atherosclerotic plaques[J].Acta Pharmaceutica Sinica B,2022,第4期
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Lei Wu1,Lingling Wang1,Xi Liu1,Yuli Bai1,Ruinan Wu1,Xiang Li1,Yutong Mao1,Ling Zhang2,Yongxiang Zheng3,Tao Gong1,Zhirong Zhang1,Yuan Huang1(Key Laboratory of Drug Targeting and Drug Delivery System,Ministry of Education,West China School of Pharmacy,Sichuan University;Sichuan University,College of Polymer Science and Engineering;Sichuan University West China School of Pharmacy).Milk-derived exosomes exhibit versatile effects for improved oral drug delivery[J].Acta Pharmaceutica Sinica B,2022,第4期
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Yuyun Tang1,Jinchao Gao1,Tao Wang2,Qian Zhang1,Antian Wang1,Meng Huang1,Renhe Yu1,Hongzhuan Chen1,3,Xiaoling Gao1(Department of Pharmacology and Chemical Biology,Shanghai Universities Collaborative Innovation Center for Translational Medicine,Shanghai Jiao Tong University School of Medicine;Department of Geriatric Psychiatry,Shanghai Mental Health Center,Shanghai Jiao Tong University School of Medicine,Alzheimer's Disease and Related Disorder Center,Shanghai Jiao Tong University;Institute of Interdisciplinary Integrative Biomedical Research,Shuguang Hospital,Shanghai University of Traditional Chinese Medicine).The effect of drug loading and multiple administration on the protein corona formation and brain delivery property of PEG-PLA nanoparticles[J].Acta Pharmaceutica Sinica B,2022,第4期
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Boyi Niu1,Yixian Zhou1,Kaixin Liao1,Ting Wen1,Sixian Lao1,Guilan Quan2,Xin Pan1,Chuanbin Wu1,2(School of Pharmaceutical Sciences,Sun Yat-sen University;College of Pharmacy,Jinan University).“Pincer movement”:Reversing cisplatin resistance based on simultaneous glutathione depletion and glutathione S-transferases inhibition by redox-responsive degradable organosilica hybrid nanoparticles[J].Acta Pharmaceutica Sinica B,2022,第4期
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Tengfei Xue1,Juan Ji1,Yuqin Sun1,Xinxin Huang2,Zhenyu Cai1,Jin Yang1,Wei Guo1,Ruobing Guo1,Hong Cheng2,Xiulan Sun1,3(Department of Pharmacology,Neuroprotective Drug Discovery Key Laboratory,Jiangsu Key Laboratory of Neurodegeneration,Nanjing Medical University;The First Affiliated Hospital of Nanjing Medical University;Nanjing University of Chinese Medicine,the Affiliated Hospital of Nanjing University of Chinese Medicine).Sphingosine-1-phosphate, a novel TREM2 ligand, promotes microglial phagocytosis to protect against ischemic brain injury[J].Acta Pharmaceutica Sinica B,2022,第4期
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Lei Feng1,2,Xiangge Tian2,Dahong Yao3,Zhenlong Yu2,Xiaokui Huo1,2,Zhenhao Tian4,Jing Ning2,Jingnan Cui4,Tony D.James5,6,Xiaochi Ma1,2(Second Affiliated Hospital,Dalian Medical University;College of Pharmacy,the National&Local Joint Engineering Research Center for Drug Development of Neurodegenerative Disease,Dalian Medical University;School of Pharmaceutical Sciences,Shenzhen Technology University;State Key Laboratory of Fine Chemicals,Dalian University of Technology;Department of Chemistry,University of Bath;School of Chemistry and Chemical Engineering,Henan Normal University).A practical strategy to develop isoform-selective near-infrared fiuorescent probes for human cytochrome P450 enzymes[J].Acta Pharmaceutica Sinica B,2022,第4期
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Chuanbin Yang1,2,Chengfu Su1,3,4,Ashok Iyaswamy1,3,Senthil Kumar Krishnamoorthi1,Zhou Zhu1,3,Sichang Yang1,Benjamin Chunkit Tong1,3,Jia Liu1,3,Sravan G.Sreenivasmurthy1,3,Xinjie Guan1,Yuxuan Kan1,Aston Jiaxi Wu1,Alexis Shiying Huang1,Jieqiong Tan5,Kingho Cheung1,3,Juxian Song1,6,Min Li1,3(Mr.&Mrs.Ko Chi-Ming Centre for Parkinson's Disease Research,School of Chinese Medicine,Hong Kong Baptist University;Department of Geriatrics,Shenzhen People's Hospital(the Second Clinical Medical College,Jinan University,the First Affiliated Hospital,Southern University of Science and Technology);Institute for Research and Continuing Education,Hong Kong Baptist University;College of Pharmacy,Henan University of Chinese Medicine;Center for Medical Genetics and Hunan Key Laboratory of Animal Model for Human Diseases,School of Life Sciences,Central South University;Medical College of Acupuncture-Moxibustion and Rehabilitation,Guangzhou University of Chinese Medicine).Celastrol enhances transcription factor EB(TFEB)-mediated autophagy and mitigates Tau pathology:Implications for Alzheimer’s disease therapy[J].Acta Pharmaceutica Sinica B,2022,第4期
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Minsong Guo1,Fengdan Zhu1,Wenqiao Qiu1,2,Gan Qiao1,Betty Yuen-Kwan Law3,Lu Yu1,Jianming Wu1,Yong Tang1,3,Chonglin Yu1,Dalian Qin1,Xiaogang Zhou1,Anguo Wu1(Sichuan Key Medical Laboratory of New Drug Discovery and Druggability Evaluation,Luzhou Key Laboratory of Activity Screening and Druggability Evaluation for Chinese Materia Medica,School of Pharmacy,Education Ministry Key Laboratory of Medical Electrophysiology,Southwest Medical University;Department of Neurosurgery Sichuan Provincial People's Hospital,University of Electronic Science and Technology of China;State Key Laboratory of Quality Research in Chinese Medicine,Macau University of Science and Technology).High-throughput screening for amyloid-β binding natural small-molecules based on the combinational use of biolayer interferometry and UHPLC-DAD-Q/TOF-MS/MS[J].Acta Pharmaceutica Sinica B,2022,第4期
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Zhiwei Zhang1,2,Suling Ding1,Zhe Wang3,Xiaowei Zhu1,Zheliang Zhou1,Weiwei Zhang1,Xiangdong Yang1,3,4,5,Junbo Ge1,3,4,5(Institutes of Biomedical Sciences and Shanghai Institute of Cardiovascular Diseases,Zhongshan Hospital,Fudan University;Reproductive Medicine Centre,Zhongshan Hospital,Fudan University;Department of Cardiology,Zhongshan Hospital,Fudan University;NHC Key Laboratory of Viral Heart Diseases,Fudan University;Key Laboratory of Viral Heart Diseases,Chinese Academy of Medical Sciences).Prmt1 upregulated by Hdc deficiency aggravates acute myocardial infarction via NETosis[J].Acta Pharmaceutica Sinica B,2022,第4期
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Rong Xiang1,Zhengsen Yu1,Yang Wang1,Lili Wang2,Shanshan Huo1,Yanbai Li1,Ruiying Liang1,Qinghong Hao1,Tianlei Ying3,Yaning Gao4,Fei Yu1,Shibo Jiang3(College of Life Sciences,Hebei Agricultural University;Research Center of Chinese Jujube,Hebei Agricultural University;Key Laboratory of Medical Molecular Virology(MOE/NHC/CAMS),School of Basic Medical Sciences,Shanghai Institute of Infectious Diseases and Biosecurity,Fudan University;Beijing Pharma and Biotech Center).Recent advances in developing small-molecule inhibitors against SARS-CoV-2[J].Acta Pharmaceutica Sinica B,2022,第4期
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Saba R.Aliyari1,Amir Ali Ghaffari1,Olivier Pernet1,2,Kislay Parvatiyar1,Yao Wang1,Hoda Gerami1,Ann-Jay Tong1,Laurent Vergnes3,Armin Takallou1,Adel Zhang1,Xiaochao Wei4,Linda D.Chilin5,Yuntao Wu5,Clay F.Semenkovich4,6,Karen Reue3,Stephen T.Smale1,Benhur Lee1,Genhong Cheng1(Department of Microbiology,Immunology and Molecular Genetics,University of California;En Viro International Laboratories;Department of Human Genetics,David Geffen School of Medicine,University of California;Division of Endocrinology,Metabolism and Lipid Research,Washington University School of Medicine;Center for Infectious Disease Research,School of Systems Biology,George Mason University Manassas;Diabetic Cardiovascular Disease Center,Washington,University School of Medicine).Suppressing fatty acid synthase by type Ⅰ interferon and chemical inhibitors as a broad spectrum anti-viral strategy against SARS-CoV-2[J].Acta Pharmaceutica Sinica B,2022,第4期
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Xueqin He1,Xiaorong Wang1,Lianyi Yang1,Zhihang Yang1,Wenqi Yu1,Yazhen Wang1,Rui Liu1,Meiwan Chen2,Huile Gao1(Key Laboratory of Drug-Targeting and Drug Delivery System of the Education Ministry and Sichuan Province,Sichuan Engineering Laboratory for Plant-Sourced Drug and Sichuan Research Center for Drug Precision Industrial Technology,West China School of Pharmacy,Sichuan University;State Key Laboratory of Quality Research in Chinese Medicine,Institute of Chinese Medical Sciences,University of Macau).Intelligent lesion blood-brain barrier targeting nano-missiles for Alzheimer’s disease treatment by anti-neuroinfiammation and neuroprotection[J].Acta Pharmaceutica Sinica B,2022,第4期
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Yongrong Yao,Huachao Chen,Ninghua Tan(State Key Laboratory of Natural Medicines,School of Traditional Chinese Pharmacy,China Pharmaceutical University).Cancer-cell-biomimetic nanoparticles systemically eliminate hypoxia tumors by synergistic chemotherapy and checkpoint blockade immunotherapy[J].Acta Pharmaceutica Sinica B,2022,第4期
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Shuai Guo,Kening Li,Yanwen Chen,Bin Li(State Key Laboratory of Natural Medicines and School of Traditional Chinese Pharmacy,China Pharmaceutical University).Unraveling the drug distribution in brain enabled by MALDI MS imaging with laser-assisted chemical transfer[J].Acta Pharmaceutica Sinica B,2022,第4期
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Yang He1,2,3,4,Yuefei Fang1,5,Meng Zhang1,6,Yuge Zhao1,Bin Tu1,2,Mingjie Shi1,Bahtiyor Muhitdinov1,7,Akmal Asrorov1,7,Qin Xu5,Yongzhuo Huang1,2,3,8(State Key Laboratory of Drug Research,Shanghai Institute of Materia Medica,Chinese Academy of Sciences;University of Chinese Academy of Sciences;Zhongshan Institute for Drug Discovery,Chinese Academy of Sciences;Department of Pharmacy,the First Affiliated Hospital of Zhengzhou University;Artemisinin Research Center,Guangzhou University of Chinese Medicine;Women's Hospital,School of Medicine,Zhejiang University;Institute of Bioorganic Chemistry,Uzbekistan Academy of Sciences;National Medical Products Administration,Key Laboratory for Quality Research and Evaluation of Pharmaceutical Excipients).Remodeling “cold” tumor immune microenvironment via epigenetic-based therapy using targeted liposomes with in situ formed albumin corona[J].Acta Pharmaceutica Sinica B,2022,第4期
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Mélanie Robert1,2,3,Bastien Laperrousaz1,Diana Piedrahita1,Emilie-Fleur Gautier3,4,Travis Nemkov5,6,Florian Dupuy4,7,Elie Nader2,3,Virginie Salnot4,Patrick Mayeux3,4,Angelo D’Alessandro5,6,Catherine Lavazec4,7,Philippe Joly2,3,8,Alexander Scheer1,Philippe Connes2,3,Agnès Cibiel1(Erytech Pharma;Laboratoire interuniversitaire de Biologie de la Motricité(LIBM)EA7424,Team?Vascular Biology and Red Blood Cell?,Université Claude Bernard Lyon 1,Université de Lyon;Labex GR-Ex;3P5 proteom’IC facility,Université de Paris,Institut Cochin,INSERM,CNRS;University of Colorado,Anschutz Medical Campus;Omix Technologies,Inc.;Inserm U1016,CNRS 8104,Université de Paris,Institut Cochin;Laboratoire de Biochimie et de Biologie Moléculaire,UF de biochimie des pathologies érythrocytaires,Centre de Biologie et de Pathologie Est,Hospices Civils de Lyon).Multiparametric characterization of red blood cell physiology after hypotonic dialysis based drug encapsulation process[J].Acta Pharmaceutica Sinica B,2022,第4期
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